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  1. 学術雑誌論文
  2. 琉球医学会
  3. 琉球医学会誌
  4. 12巻4号
  1. 部局別インデックス
  2. その他

[原著]リドカイン代謝に及ぼすブピバカインの影響 : in vitro, in vivo での検討

http://hdl.handle.net/20.500.12000/0002015920
http://hdl.handle.net/20.500.12000/0002015920
cd75e241-ac25-427a-a7bf-8263ddf858c4
名前 / ファイル ライセンス アクション
v12p375.pdf v12p375.pdf
Item type デフォルトアイテムタイプ(フル)(1)
公開日 2010-07-02
タイトル
タイトル [原著]リドカイン代謝に及ぼすブピバカインの影響 : in vitro, in vivo での検討
言語 ja
作成者 磯, 淳典

× 磯, 淳典

ja 磯, 淳典

平良, 豊

× 平良, 豊

ja 平良, 豊

垣花, 脩

× 垣花, 脩

ja 垣花, 脩

濱田, 哲

× 濱田, 哲

ja 濱田, 哲

奥田, 佳朗

× 奥田, 佳朗

ja 奥田, 佳朗

Iso, Atunori

× Iso, Atunori

en Iso, Atunori

Taira, Yutaka

× Taira, Yutaka

en Taira, Yutaka

Kakinohana, Osamu

× Kakinohana, Osamu

en Kakinohana, Osamu

Hamada, Satosi

× Hamada, Satosi

en Hamada, Satosi

Okuda, Yoshiaki

× Okuda, Yoshiaki

en Okuda, Yoshiaki

アクセス権
アクセス権 open access
アクセス権URI http://purl.org/coar/access_right/c_abf2
権利情報
言語 ja
権利情報 琉球医学会
主題
言語 en
主題Scheme Other
主題 biotransformation
言語 en
主題Scheme Other
主題 pharmacokinetics
言語 en
主題Scheme Other
主題 enzyme inhibition
言語 en
主題Scheme Other
主題 lidocain
言語 en
主題Scheme Other
主題 bupivacaine
内容記述
内容記述タイプ Other
内容記述 To evaluate the effects of bupivacaine on lidocaine metabolism mediated by chtochrome P-450, we analyzed enzyme kinetics in an in vitro study using rat liver microsomes and pharmacokinetics in an in vivo study using anesthetized dogs. In vitro study,bupivacaine showed mixed type inhibition of hdocaine metabolism with inhibition constants being 1.38mM. Since bupivacaine did not affect cytochrome C reductase activity,this inhibition of lidocaine metabolism may have been caused by the action on cytochrome P-450. In vivo study, there was no difference between pharmacokinetic parameter after lidocaine alone injection and lidocaine mixed with bupivacaine injection.
内容記述タイプ Other
内容記述 論文
出版者
言語 ja
出版者 琉球医学会
言語
言語 jpn
資源タイプ
資源タイプ journal article
資源タイプ識別子 http://purl.org/coar/resource_type/c_6501
出版タイプ
出版タイプ VoR
出版タイプResource http://purl.org/coar/version/c_970fb48d4fbd8a85
収録物識別子
収録物識別子タイプ ISSN
収録物識別子 1346888X
収録物識別子タイプ ISSN
収録物識別子 0289-1530
収録物識別子タイプ NCID
収録物識別子 AN10369445
収録物名
言語 ja
収録物名 琉球医学会誌 = Ryukyu Medical Journal
書誌情報
巻 12, 号 4, p. 375-382
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